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- Carbamazepine has also been shown to potentiate GABA receptors made up of alpha1, beta2, gamma2 subunits.<ref>Granger, P. et al. Modulati16 KB (2,164 words) - 16:42, 27 September 2010
- ...eceptors in the absence of the GABA molecule, whereas benzodiazepines need GABA to be present to have an effect: this may explain the more widespread effec ...0.1038/sj.bjp.0705942 | pmc = 1575970}}</ref> Such findings implicate (non-GABA-ergic) ligand-gated ion channels, e.g. the neuronal nAChR channel, in media24 KB (3,339 words) - 16:46, 27 September 2010
- ...trations, but not α<sub>1</sub>β<sub>2</sub>γ<sub>2</sub> receptors.<ref name="Korpi95"/><ref name="Wafford96"/> During development, the &alpha12 KB (1,678 words) - 16:48, 27 September 2010
- ...or|5-HT<sub>3</sub> receptor]]s, and slightly potentiates [[GABAA receptor|GABA<sub>A</sub>]] and [[glycine receptor]]s.<ref name="pmid11020766">{{cite jou ...ytic effect in mice in the elevated plus maze: mediation by benzodiazepine receptors|author = Emmanouil, D.E., Johnson, C.H. & Quock, R.M.|journal = Psychopharm61 KB (8,728 words) - 16:50, 27 September 2010
- ...smitter GABA by binding to the benzodiazepine site on the [[GABAA receptor|GABA<sub>A</sub> receptor]] leading to [[central nervous system]] depression.<re ...ing-2006">{{Cite journal | last1 = Whiting | first1 = PJ. | title = GABA-A receptors: a viable target for novel anxiolytics? | journal = Curr Opin Pharmacol | v78 KB (10,295 words) - 16:51, 27 September 2010
- .... [http://www.nature.com/bjp/journal/v143/n4/full/0705974a.html "Selective GABA-receptor actions of amobarbital on thalamic neurons."] ''British Journal of9 KB (1,128 words) - 22:04, 21 September 2010
- ...ally diverse class of mostly synthetic substances that bind to cannabinoid receptors. The latter group encompasses a variety of distinct chemical classes: the ' == Cannabinoid receptors ==49 KB (6,487 words) - 22:06, 21 September 2010
- ...tin''') is a pharmaceutical drug, specifically a [[gamma-Aminobutyric acid|GABA]] [[Analogue (chemistry)|analogue]]. It was originally developed for the tr ...inobutyric acid ('''GABA'''), but is not believed to act on the same brain receptors.30 KB (4,025 words) - 22:06, 21 September 2010
- ...5 |pmc=430630}}</ref> what Eric Simon (who independently discovered opioid receptors in the brain) later termed "endorphin" by an [[abbreviation]] of "endogenou ...gastric and vascular function as well as possibly panic and satiation, and receptors are often found at postsynaptic locations as well as presynaptically.18 KB (2,467 words) - 22:06, 21 September 2010
- ...ocannabinoid noladin ether acts as a full agonist at human CB2 cannabinoid receptors }}</ref> It shows agonistic behaviour on both receptors and is a partial agonist for the [[TRPV1]] channel.<ref name="pmid15148262"6 KB (807 words) - 22:08, 21 September 2010
- ...st. In addition, oleamide potentiates several serotonin receptors and the GABA(A) receptor, and inhibits gap junction communication.5 KB (687 words) - 22:09, 21 September 2010
- ...beta, gamma or delta subunits (some consist of 5 alpha subunits). Cys-loop receptors possess a characteristic loop formed by a disulfide bond between two [[cyst ...l | author = Albuquerque et al | title = Mammalian Nicotinic Acetylcholine Receptors: from Structure to Function | journal = Physiol Rev| issue = 89| pages = 732 KB (312 words) - 22:11, 21 September 2010
- ...r case the receptors are typically 7-membrane spanning [[G-protein coupled receptors]] while in the latter case they are [[ligand-gated ion channels]]. The form Most other neurotransmitters, on the other hand, e.g. [[glutamate]], [[GABA]] and [[glycine]], are used very generally throughout the central nervous s11 KB (1,374 words) - 22:11, 21 September 2010
- ...the activity of K<sub>Ca</sub>2.3 channels on the [[cell membrane]]. In [[GABA]]ergic [[POA neurons]], estrogen enhanced the ability of [[alpha-1 adrenerg14 KB (1,907 words) - 22:12, 21 September 2010
- ...journal |author=Vicini S |title=New perspectives in the functional role of GABA(A) channel heterogeneity |journal=Mol. Neurobiol. |volume=19 |issue=2 |page ...ided into 6 subfamilies based on homology: classical ([[TRPC]]), vanilloid receptors ([[TRPV]]), melastatin ([[TRPM]]), polycystins ([[TRPP]]), mucolipins ([[TR31 KB (4,177 words) - 22:12, 21 September 2010
- .../sup>]], [[calcium|Ca<sup>2+</sup>]], or [[chloride|Cl<sup>-</sup>]]. Such receptors located at [[synapse]]s convert the chemical signal of [[presynaptic]]ally ...= Structure and function of the glycine receptor and related nicotinicoid receptors | journal = J. Biol. Chem. | volume = 279 | issue = 19 | pages = 19383–617 KB (2,344 words) - 22:12, 21 September 2010
- ...etomidate and propofol at beta3-containing gamma-aminobutyric acid type A receptors. ''Neuropharmacology''. 2009 Sep;57(4):446-55. PMID 19555700</ref>10 KB (1,350 words) - 21:01, 24 September 2010
- ...ich is associated with Cl<sup>−</sup> [[ionophore]]s at GABA<sub>A</sub> receptors.<ref>Katzung, Bertram G., Basic and Clinical Pharmacology, 10th ed., p. 4063 KB (345 words) - 21:01, 24 September 2010
- ...propofol analogues: mapping binding sites for an anesthetic phenol on the GABA(A) receptor. ''Journal of Medicinal Chemistry''. 2002 Jul 18;45(15):3210–21 KB (2,875 words) - 21:03, 24 September 2010
- ...[[Henri Laborit]] to use in studying the neurotransmitter [[GABA receptor|GABA]].<ref>{{cite journal | author = H. Laborit, J.M. Jouany, J. Gerald, F. Fab .../pjp/pdf/2004/1_43.pdf|format=PDF}}</ref> GHB is probably synthesized from GABA in GABAergic [[neurons]], and released when the neurons fire.<ref name="mec55 KB (7,839 words) - 21:04, 24 September 2010