4-Phenylfentanyl

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4-Phenylfentanyl
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Systematic (IUPAC) name
N-(1-phenethyl-4-phenyl-4-piperidyl)-N-phenyl-propanamide
Identifiers
ATC code none
PubChem CID 10319503
Synonyms 4-Phenylfentanyl
Chemical data
Formula C28H32N2O
Molar mass 412.565 g/mol[[Script error: No such module "String".]]
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4-Phenylfentanyl is an opioid analgesic that is a derivative of fentanyl. It was developed during the course of research that ultimately resulted in super-potent opioid derivatives such as carfentanil, though it is a substantially less potent analogue. 4-Phenylfentanyl is around 8x the potency of fentanyl in analgesic tests on animals, but more complex 4-heteroaryl derivatives such as substituted thiophenes and thiazoles are more potent still, as they are closer bioisosteres to the 4-carbomethoxy group of carfentanil.[1]

Side effects of fentanyl analogues are similar to those of fentanyl, and include itching, nausea and potentially serious respiratory depression which can be life-threatening.

References

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