Lesopitron

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Lesopitron
File:Lesopitron.png
Systematic (IUPAC) name
2-{4-[4-(4-chloro-1H-pyrazol-1-yl)butyl]piperazin-1-yl}pyrimidine
Clinical data
Routes of
administration
Oral
Legal status
Legal status
  • Uncontrolled
Identifiers
CAS Number 132449-46-8
ATC code none
PubChem CID 60813
ChemSpider 54801
Chemical data
Formula C15H21ClN6
Molar mass 320.82 g/mol[[Script error: No such module "String".]]
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Lesopitron (E-4424) is a selective full agonist of the 5-HT1A receptor which is structurally related to the azapirones.[1] In 2001 it was under development by Esteve as an anxiolytic for the treatment of generalized anxiety disorder (GAD).[2][3] It made it to phase II clinical trials but was apparently discontinued as no new information on lesopitron has surfaced since.[2][3]

See also

References

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