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...iate receptor sites within the CNS (a competitive antagonist, not a direct agonist), thereby preventing the action of both [[endogenous]] and [[xenobiotic]] o ...e nasal [[mucosa]].<ref name="pmid15039670">{{cite journal |vauthors=Wolfe TR, Bernstone T | title = Intranasal drug delivery: an alternative to intraven

...[[Chugai Pharmaceuticals]] discovered an erythromycin-derived [[motilin]] agonist called [[Mitemcinal]] that is believed to have strong [[prokinetic]] proper ...>{{cite journal |author=Weber FH Jr, et. al |title=Erythromycin: a motilin agonist and gastrointestinal prokinetic agent |journal=American Journal of Gastroen

...-acting [[cholinergic]] antagonist) or [[phenylephrine]] (an α-adrenergic agonist) is preferred as an aid to [[ophthalmic]] examination. Atropine induces [[m [[tr:Atropin]]

...cker MW, Brioni JD, Moreland RB, Fox GB. A-412997, a selective dopamine D4 agonist, improves cognitive performance in rats. ''Pharmacology, Biochemistry and B ...[spinal cord]],<ref>Jensen TS, Yaksh TL.Effects of an intrathecal dopamine agonist, apomorphine, on thermal and chemical evoked noxious responses in rats.Brai

...and Type II receptor agonist), or [[RU28362]] (a specific Type II receptor agonist), to adrenalectomized animals induced changes in [[leukocyte distribution]] [[tr:Kortizol]]

[[tr:Adrenalin]]

...ids differ in the intensity and length of each, and weak opioids and mixed agonist-antagonists may have acute withdrawal syndromes which do not reach the high ...tor|&kappa;-opioid]] and [[delta opioid receptor|&delta;-opioid]] receptor agonist, κ-opioid's action is associated with spinal analgesia, [[miosis]] (pinpoi

...is an [[Alpha-1 adrenergic receptor|α₁-adrenergic receptor]] [[agonist]] used primarily as a [[decongestant]], as an agent to dilate the [[pupil]] ...ref>. Because phenylephrine is a direct selective α-adrenergic [[receptor agonist]], it does not cause the release of endogenous [[Norepinephrine|noradrenali

* Adenocard - Adenosine agonist, primarily used as an anti-[[arrhythmia|arrhythmic]]. [[tr:Vazodilatör]]

...ntification of two related pentapeptides from the brain with potent opiate agonist activity |journal=Nature |volume=258 |issue=5536 |pages=577–80 |year=1975 ...ker ME, Henriksen G, Koppenhoefer M, Wagner KJ, Valet M, Berthele A, Tolle TR | title = The Runner's High: Opioidergic Mechanisms in the Human Brain | jo

...]] system. [[Tramadol]] and [[buprenorphine]] are thought to be [[partial agonist]]s of the opioid receptors.{{Citation needed|reason=tramadol|date=February [[tr:Analjezik]]

...aker JL, Seely KA, Reed RL, Crow JP, Prather PL |title=The CB2 cannabinoid agonist AM-1241 prolongs survival in a transgenic mouse model of amyotrophic latera

'''Tetrahydrocannabinol''' ({{pron-en|ˌtɛtrəˌhaɪdrɵkəˈnæbɨnɒl}} {{Respell|tet-rə|HYE|drə-kə|NAB|i-nol}}) (' ..., mainly present in cells of the [[immune system]]. It acts as a partial [[agonist]] on both receptors, i.e., it activates them but not to their full extent.

...date= |accessdate=2010-07-28}}</ref> In addition, it is a synthetic strong agonist at the [[mu opioid receptor|μ-opioid]] receptors. Historically it has been [[tr:Fentanil]]

Methadone is a full µ-opioid [[agonist]]. Methadone also binds to the glutamatergic [[NMDA]] (N-methyl-D-aspartate [[tr:Methadon]]

...al]];<ref name="Zhang2005pabs" /><ref name="Valdés1983" /> as a κ-opioid agonist. ...it is an even more potent [[D2 receptor|D₂ receptor]] [[partial agonist]], and it is likely this action plays a significant role in its effects as