Ciclotizolam

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Ciclotizolam
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Systematic (IUPAC) name
2-Bromo-4-(o-chlorophenyl)-9-cyclohexyl-6H-thieno(3,2-f)-s-triazolo(4,3-a)(1,4)diazepine
Identifiers
CAS Number 58765-21-2
ATC code none
PubChem CID 71949
ChemSpider 64956
Chemical data
Formula C20H18BrClN4S
Molar mass 461.806[[Script error: No such module "String".]]
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Ciclotizolam (WE-973) is a drug which is a thienobenzodiazepine derivative. It is a partial agonist for the benzodiazepine site of the GABAA receptor, with similar binding affinity to related compounds like brotizolam, but a low efficacy.[1][2]

See also

References

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  2. Ikeda M, Weber KH, Bechtel WD, Malatynska E, Yamamura HI (1989). "Relative efficacies of 1,4-diazepines on GABA-stimulated chloride influx in rat brain vesicles". Life Sciences. 45 (4): 349–58. doi:10.1016/0024-3205(89)90145-8. PMID 2569655.