GR-89696
From Self-sufficiency
Revision as of 20:50, 29 July 2010 by PotatoBot (Talk) (Stub sorting and placement of stub template(s): analgesic-stub)
200px | |
Systematic (IUPAC) name | |
---|---|
methyl 4-[2-(3,4-dichlorophenyl)acetyl]-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate | |
Identifiers | |
CAS Number | 126766-32-3 |
PubChem | CID 3505 |
Chemical data | |
Formula | C19H25Cl2N3O3 |
Molar mass | 414.325 g/mol[[Script error: No such module "String".]] |
Script error: No such module "collapsible list". |
GR-89696 is a drug which acts as a highly selective κ-opioid agonist.[1] It shows selective effects in different animal models and it is thought it may be a subtype-selective agonist for the κ2 subtype.[2][3][4] Recent studies have suggested that GR-89696 and related κ2-selective agonists may be useful for preventing the itching which is a common side effect of conventional opioid analgesic drugs, without the additional side effects of non-selective kappa agonists.[5]
References
- ↑ Lua error in package.lua at line 80: module 'Module:Citation/CS1/Suggestions' not found.
- ↑ Lua error in package.lua at line 80: module 'Module:Citation/CS1/Suggestions' not found.
- ↑ Lua error in package.lua at line 80: module 'Module:Citation/CS1/Suggestions' not found.
- ↑ Lua error in package.lua at line 80: module 'Module:Citation/CS1/Suggestions' not found.
- ↑ Lua error in package.lua at line 80: module 'Module:Citation/CS1/Suggestions' not found.
40px | This analgesic-related article is a stub. You can help ssf by expanding it. |
Categories:
- Pages with script errors
- Pages with broken file links
- Infobox drug tracked parameters
- Articles without EBI source
- Chemical pages without ChemSpiderID
- Chemical pages without DrugBank identifier
- Articles without KEGG source
- Articles without InChI source
- Articles without UNII source
- Drugboxes with an unspecified ATC code
- Drugs with no legal status
- Articles containing unverified chemical infoboxes
- Opioids
- Organochlorides
- Acetamides
- Piperazines
- Pyrrolidines
- Kappa agonists
- Analgesic stubs
- 2Fix