Befiradol

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Befiradol
File:F-13640 structure.png
Systematic (IUPAC) name
3-​chloro-​4-​fluorophenyl-​[4-​fluoro-​4-​([(5-​methylpyridin-​2-yl)methylamino]methyl)piperidin-​1-​yl]methanone
Legal status
Legal status
  • Uncontrolled
Identifiers
CAS Number 208110-64-9
ATC code none
PubChem CID 9865384
Chemical data
Formula C20H22Cl1F2N3O1
Molar mass 393.857 g/mol
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Befiradol (F-13,640) is a very potent and highly selective 5-HT1A receptor full agonist. It has powerful analgesic and antiallodynic effects comparable to those of high doses of opioid painkillers, but with fewer and less prominent side effects, as well as little or no development of tolerance with repeated use.[1][2][3][4][5][6]

See also

References

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Opioids
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Propionic acid class
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Anthranilic acid
(fenamate) class
Atypical, Adjuvant & Potentiators,
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α2δ VDCC Blockers
5-HT1A Agonists
Azapirones: Buspirone • Gepirone • Tandospirone; Others: Flesinoxan • Oxaflozane
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Diphenylmethanes: Captodiame • Hydroxyzine; Others: Brompheniramine • Chlorpheniramine • Pheniramine
CRH1 Antagonists
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mGluR5 NAMs
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  6. ↑ Bernard Vacher, Bernard Bonnaud, Wouter Koek. Pyridin-2-yl-methylamine derivatives, method of preparing and application as medicine. US Patent 6020345, May 21, 1999.
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